Angiotensin Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB01062 | Valsartan | 137862-53-4 | Valsartan is a selective angiotensin II AT1 receptor antagonist with elimination half-life of 6 hours. |
| FB08896 | trans-Tranilast | 70806-55-2 | trans-Tranilast is an antiallergic drug, used to treat bronchial asthma, allergic rhinitis and atopic dermatitis. |
| FB01967 | Tranilast Sodium | 104931-56-8 | Tranilast is an antiallergic agent. |
| FB00297 | Tranilast | 53902-12-8 | Tranilast can antagonize angiotensin II and also work as an antiallergic agent. |
| FB01510 | Telmisartan | 144701-48-4 | Telmisartan is an angiotensin II receptor antagonist with Ki value of 3.7nM, used in the management of hypertension with elimination half-life of 24 hours. |
| FB09672 | Tasosartan | 145733-36-4 | Tasosartan is a long-acting angiotensin II receptor blocker. |
| FB11693 | SL910102 | 144756-71-8 | SL910102 is a nonpeptide angiotensin AT1 receptor antagonist. |
| FB01222 | PD123319 Ditrifluoroacetate | 136676-91-0 | PD123319 Ditrifluoroacetate is a potent, selective and non-peptide angiotensin AT2 receptor antagonist. |
| FB08036 | PD123319 | 130663-39-7 | PD 123319 is a potent, selective AT2 angiotensin II receptor antagonist with IC50 of 34 nM. |
| FB01509 | Olmesartan Medoxomil | 144689-63-4 | Olmesartan Medoxomil is a synthetic imidazole-derived angiotensin II receptor antagonist, acting as a prodrug with an antihypertensive property. |
| FB07832 | Olmesartan | 144689-24-7 | Olmesartan is an antagonist of angiotensin II receptor, working as an antihypertensive agent. |
| FB09765 | Losartan Potassium | 124750-99-8 | Losartan Potassium is the potassium salt form of Losartan, which is a compeitive AT1 receptor inhibitor with IC50 value of 20 nM. |
| FB10642 | Losartan | 114798-26-4 | Losartan is a compeitive AT1 receptor inhibitor with IC50 value of 20 nM. |
| FB01939 | Losartan D4 | 1030937-27-9 | Losartan D4 is deuterium labeled Losartan, which is an angiotensin II receptor antagonist. |
| FB00682 | LCZ 696 | 936623-90-4 | LCZ 696 is a mixture of neprilysin inhibitor sacubitril and the angiotensin receptor blocker valsartan in a ratio of 1:1. |
| FB01103 | Irbesartan | 138402-11-6 | Irbesartan is a selective and competitive nonpeptide angiotensin II antagonist with antihypertensive activity. |
| FB09247 | Fimasartan | 247257-48-3 | Fimasartan is an improved non-peptide angiotensin II receptor blocker used for the treatment of hypertension and heart failure, which enables higher potency and longer duration than losartan. |
| FB01326 | Eprosartan Mesylate | 144143-96-4 | Eprosartan Mesylate is a reversible and competitive angiotensin II receptor inhibitor. |
| FB01325 | Eprosartan | 133040-01-4 | Eprosartan is an angiotensin II receptor antagonist used for the treatment of high blood pressure. |
| FB09971 | EMA401 | 1316755-16-4 | EMA401, a highly selective AT2R antagonist, inhibition of augmented AngII/AT2R induced p38 and p42/p44 MAPK activation, and hence inhibition of DRG neuron hyperexcitability and sprouting of DRG neurons. |
| FB02699 | CGP-42112 | 127060-75-7 | CGP-42112 is a potent Angiotensin-II subtype 2 receptor (AT2 R) agonist. |
| FB01211 | Candesartan | 139481-59-7 | Candesartan is a benzimidazole-derived and competitive AT1 inhibitor with IC50 value of 0.26 nM. |
| FB01606 | Candesartan Cilexetil | 145040-37-5 | Candesartan Cilexetil is a benzimidazole-derived and competitive AT1 inhibitor with IC50 value of 0.26 nM. |
| FB02744 | BIBS 39 | 133085-33-3 | BIBS 39 is a nonpeptide angiotensin II (AII) receptor antagonist. |
| FB02563 | Azilsartan Medoxomil | 863031-21-4 | Azilsartan Medoxomil is an orally available angiotensin II type 1 (AT1) receptor antagonist with IC50 value of 2.6 nM. |
| FB02194 | Azilsartan Medoxomil Potassium | 863031-24-7 | Azilsartan medoxomil is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. |
| FB07915 | Azilsartan | 147403-03-0 | Azilsartan is an orally available angiotensin II type 1 (AT1) receptor antagonist with IC50 value of 2.6 nM. |
| FB01523 | AVE 0991 Sodium | 306288-04-0 | AVE 0991 sodium is a nonpeptide Ang-(1-7) receptor Mas agonist, represents an important step for exploration of the effects of Ang-(1-7) and testing of its potential as a cardiovascular drug. |
| FB01087 | AVE 0991 | 304462-19-9 | AVE 0991 is a nonpeptide Ang-(1-7) receptor Mas agonist. |
| FB11227 | AT2R Agonist C21 | 477775-14-7 | AT2R agonist C21 is a small-molecule ATR receptor (AT2R) agonist. |
| FB10627 | Angiotensin II | 4474-91-3 | Angiotensin II human is a peptide hormone that causes vasoconstriction and a subsequent increase in blood pressure. |
| FB04606 | Angiotensin II 5-Valine | 58-49-1 | Angiotensin II 5-valine is an angiotensin II analog which is an agonist at angiotensin receptors. |
| FB07742 | Angiotensin II (3-8), Human | 12676-15-2 | Angiotensin II (3-8), human is an agonist of angiotensin AT1 receptor. Its activation is relatively weak. |
| FB07702 | AHU-377 | 149709-62-6 | AHU-377 and valsartan can compose LCZ696 in a 1:1 molar ratio. It also works as an inhibitor of neprilysin with IC50 value of 5 nM. |
| FB16567 | ZD 7155 HCl | 146709-78-6 |