Kainate receptors, or kainic acid receptors (KARs), are ionotropic receptors that respond to the neurotransmitter glutamate.
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB12721 | UBP 282 | 544697-47-4 | UBP-282 is an α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) and kainate receptor antagonist. |
| FB15921 | UBP 310 | 902464-46-4 | UBP 310 is an antagonist of GluK1 (formerly GLUK5) kainate receptor with IC50 of 130 nM. |
| FB15922 | (S)-2-((3-(2-Amino-2-carboxyethyl)-2,6-dioxo-2,3-dihydropyrimidin-1(6H)-yl)methyl)benzoic acid | 745055-91-8 | UBP 302 is a potent and selective GluK1 (formally GluR5)-subunit containing kainate receptor antagonist with KD of 402 nM. |
| FB11073 | Selurampanel | 912574-69-7 | Selurampanel is a competitive AMPA/kainate receptor antagonist drug for epilepsy. |
| FB20337 | Domoic acid | 14277-97-5 | Potent and selective kainate agonist. |
| FB00609 | L-Theanine | 3081-61-6 | L-theanine is an amino acid found most commonly in tea leaves and binds to ionotropic glutamate receptors in the micromolar range, including the AMPA and kainate receptors and, to a lesser extent, the NMDA receptor. |
| FB03094 | Kainic Acid | 487-79-6 | Kainic acid is a selective agonist at kainate receptors. Potent excitant and neurotoxin. |
| FB12204 | CNQX Disodium Salt | 479347-85-8 | CNQX Disodium Salt is a AMPA/kainate antagonist and also available as part of the Kainate Receptor. |
| FB15930 | ATPA | 140158-50-5 | ATPA is a selective and potent GluK1 kainate receptor agonist with Ki of 4.3 nM. |
| FB09136 | (S)-Willardiine | 21416-43-3 | (S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 μM. |