货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
FB15526 | RTI-13951-33 | 2244884-08-8 | RTI-13951-33 is a potent, selective, and brain-penetrant GPR88 agonist, with an EC50 of 25 nM in GPR88 cAMP functional assay. RTI-13951-33 reduces alcohol reinforcement and intake behaviors in rats[1]. |
FB11567 | 2-PCCA | 1984859-71-3 | 2-PCCA is a racemic form of the GPR88 agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells. |
FB11569 | 2-PCCA HCl | N/A | 2-PCCA HCl is a GPR88 agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells. |
FB11571 | (1S,2S)-2-PCCA | 1609624-97-6 | (1S,2S)-2-PCCA is a less active diastereomer of 2-PCCA. 2-PCCA is a GPR88 agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells. |
FB11591 | (1S,2S)-2-PCCA HCl | 1609563-70-3 | (1S,2S)-2-PCCA HCl is a less active diastereomer of 2-PCCA. 2-PCCA is a GPR88 agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells. |
FB11570 | (1R,2R)-2-PCCA | 1287205-42-8 | (1R,2R)-2-PCCA is a diastereomer of 2-PCCA, and acts as a potent GPR88 agonist, with an EC50 of 3 nM. |
FB11592 | (1R,2R)-2-PCCA 2HCl | 1609563-71-4 | (1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 agonist, with an EC50 of 3 nM. |