Neurotensin Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB11322 | SR48692 | 146362-70-1 | SR48692 is an orally available neurotensin antagonist; selective for NTS1 over NTS2 (apparent affinity, Ke, is 36 nM for NTS1), and competitively inhibits binding of [125I]-neurotensin to HT29 and N1E115 cell membranes (IC50 values are 15.3 and 20.4 nM respectively). |
| FB10810 | PD149163 | 169528-11-4 | PD149163, a neurotensin receptor 1 agonist, decreases methamphetamine self-administration in DBA/2J mice without causing excessive sedation. |
| FB16513 | NEurotensin(8-13) | 60482-95-3 | Neurotensin Fragment 8-13 is the smallest active fragment of neurotensin which is a potent cellular mitogen for various colorectal and pancreatic cancers which possess high-affinity neurotensin receptors (NTR). |
| FB03245 | ML314 | 1448895-09-7 | ML314 is a potent molecule agonist of NTR1 (EC50 = 1.9 μM) and shows good selectivity against NTR2 and GPR35, but did not stimulate Ca2+ mobilization. |
| FB12326 | JMV 449 | 139026-66-7 | JMV 449 is a potent, metabolically stable neurotensin receptor agonist peptide. |