GNRH Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB00592 | Triptorelin | 57773-63-4 | Triptorelin, a GnRH agaonist, inhibits the proliferation of estradiol-induced cancer cells. |
| FB02996 | Relugolix | 737789-87-6 | Relugolix is a non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum. It possesses higher affinity and potent antagonistic activity compared with TAK-013. |
| FB07135 | Nafarelin | 76932-56-4 | Nafarelin is an agonist of gonadotropin-releasing hormone (GnRH) and can induce secretion of luteinizing hormone (LH) and follicle-stimulating hormone (FSH). |
| FB03383 | Leuprorelin | 53714-56-0 | Leuprolide is an agonist of GnRH receptors. |
| FB03773 | Leuprolide Acetate | 74381-53-6 | Leuprolide acetate, an analog of GnRH, can act as agonist of GnRH receptors. |
| FB03369 | Lecirelin | 61012-19-9 | Lecirelin is a synthetic GnRH analogue which showed a great efficacy in the treatment of bovine ovarian follicular cysts. |
| FB10713 | Goserelin | 65807-02-5 | Goserelin is an injectable gonadotropin releasing hormone superagonist (GnRH agonist). |
| FB10729 | Goserelin Acetate | 145781-92-6 | Goserelin acetate is an injectable gonadotropin releasing hormone superagonist (GnRH agonist). |
| FB03826 | Gonadorelin Acetate | 34973-08-5 | Gonadorelin acetate is a man-made protein that is like a hormone in the body called gonadotropin-releasing hormone (GnRH). |
| FB02980 | Elagolix Sodium | 832720-36-2 | Elagolix sodium is an antagonist of human GnRH receptor (GnRHR) with IC50 and Ki of 0.25 nM and 3.7 nM, respectively. |
| FB06305 | Elagolix | 834153-87-6 | Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). |
| FB00327 | Deslorelin | 57773-65-6 | Deslorelin is a GnRH agonist. |
| FB04085 | Degarelix | 214766-78-6 | Degarelix is a gonadotrophin-releasing hormone (GnRH) antagonist for the first-line treatment of androgen-dependent advanced prostate cancer. |
| FB12160 | Cetrorelix acetate(1:2) | 130143-01-0 | Cetrorelix acetate(1:2) is the acetate form of cetrorelix which is an antagonist of gonadotropin-releasing hormone (GnRH) used in inhibiting premature luteinizing hormone surges. |
| FB10298 | Cetrorelix Acetate | 145672-81-7 | Cetrorelix acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with IC50 of 1.21 nM. |
| FB10290 | Buserelin Acetate | 68630-75-1 | Buserelin acetate is a gonadotropin-releasing hormone agonist (GnRH agonist). |
| FB08777 | Alarelin Acetate | 79561-22-1 | Alarelin acetate is a synthetic agonist of GnRH. |
| FB11136 | AEZS-108 | 139570-93-7 | AEZS-108 is a peptide agonist of the gonadotropin releasing hormone-1 receptor (GnRH-1R). |
| FB07187 | Abarelix | 183552-38-7 | Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, used for prostate cancer treatment. |