Glucokinase
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB04871 | Ro 28-1675 | 300353-13-3 | Ro 28-1675 is a potent allosteric GK activator with a SC1.5 value of 0.24± 0.0019 μM. |
| FB11858 | PF-04991532 | 1215197-37-7 | PF-04991532 is a potent, hepatoselective glucokinase activator with EC50s of 80 and 100 nM in human and rat, respectively. |
| FB06555 | LY2608204 | 1234703-40-2 | LY2608204 is an activator of glucokinase (GK) with EC50 of 42 nM. |
| FB12256 | GKA 50 | 851884-87-2 | GKA 50 is a potent glucokinase activator with EC50 of 33 nM. |
| FB00040 | Dorzagliatin | 1191995-00-2 | Dorzagliatin is a glucokinase activator on glucose metabolism. |
| FB11521 | AMG-3969 | 1361224-53-4 | AMG-3969 is a glucokinase-GKRP disruptor with IC50 value of 343nM and potently reverses the inhibitory effect of GKRP on GK activity. |
| FB10346 | AM-2394 | 1442684-77-6 | AM-2394 is a structurally distinct glucokinase activator (GKA). AM-2394 activates glucokinase (GK) with an EC50 of 60 nM. |