GHSR
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB15784 | Ipamorelin | 170851-70-4 | Ipamorelin, also known as NNC-26-0161, is a a ghrelin mimetic. Ipamorelin counteracts glucocorticoid-induced decrease in bone formation of adult rats. Ipamorelin may ameliorate the symptoms in patients with POI. Ipamorelin accelerates gastric emptying in a rodent model of postoperative ileus through the stimulation of gastric contractility by activating a ghrelin receptor-mediated mechanism involving cholinergic excitatory neurons. |
| FB00959 | Ibutamoren Mesylate | 159752-10-0 | Ibutamoren mesylate is an agonist of nonpeptide growth hormone secretagogue receptor. |
| FB02497 | Examorelin | 140703-51-1 | Examorelin is a selective agonist of the ghrelin/growth hormone secretagogue receptor (GHSR). |
| FB11603 | Capromorelin Tartrate | 193273-69-7 | Capromorelin is a growth hormone secretagogue and ghrelin mimetic (hGHS-R1a Ki=7nM). Capromorelin stimulates GH release in rat pituitary cell cultures with EC50 of 3 nM |
| FB04837 | Anamorelin | 249921-19-5 | Anamorelin is a ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay. |
| FB06856 | Anamorelin HCl | 861998-00-7 | Anamorelin HCl is a synthetic orally active ghrelin receptor agonist which is under development for the management of non-small lung cancer associated cachexia/anorexia. |
| FB04908 | Anamorelin Fumarate | 339539-92-3 | Anamorelin fumarate is a ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay. |
| FB10301 | Alexamorelin | N/A | Alexamorelin is a synthetic heptapeptide which inhibits GHS binding in vitro. |