Bombesin Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB11749 | PD176252 | 204067-01-6 | PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells. |
| FB15685 | ML-18 | 1422269-30-4 | ML-18 is a nonpeptide BRS-3 antagonist with IC50 value of 4.8μM. |
| FB01933 | MK-5046 | 1022152-70-0 | MK-5046 is a BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM). |
| FB16024 | BA 1 | 183241-31-8 | BA 1 is a specific agonist of bombesin receptor with IC50 values of 0.26, 1.55 and 2.52 nM for BB1, BB2 and BB3 respectively. It can enhance glucose transport in obese and diabetic primary myocytes. |