DDR1/DDR2 Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB16506 | VU6015929 | 2442597-56-8 | VU6015929 is a potent, selective and orally active dual discoidin domain receptor 1/2 (DDR1/2) inhibitor with IC50 values of 4.67 nM and 7.39 nM, respectively and potently blocks collagen-induced DDR1 activation and collagen-IV production. |
| FB16384 | ODM-203 | 1430723-35-5 | ODM-203 is a selective inhibitor of FGFR and VEGFR with IC50 values of 11, 16, 6, 35nM for recombinant FGFR1-4 and 26, 9, 5nM for VEGFR1-3, respectively. |
| FB09615 | DDR1-IN-3 | 1934246-19-1 | DDR1-IN-3 is a selective Discoidin Domain Receptor 1 (DDR1) inhibitor, with an IC50 value of 9.4 nM. |
| FB01484 | DDR1-IN-2 | 1429617-90-2 | DDR1-IN-2 is an inhibitor of discoidin domain receptor 1 (DDR1) with IC50 of 13.1 nM, the IC50 of DDR2 is 203 nM. |
| FB03248 | DDR1-IN-1 | 1449685-96-4 | DDR1-IN-1 is a potent and selective DDR1 receptor tyrosine kinase inhibitor with IC50/EC50 of 105 nM/87 nM and 4-fold less potent for DDR2 (IC50= 413 nM). |
| FB11830 | DDR Inhibitor | 1644069-80-6 | DDR Inhibitor is a potent discoidin domain receptor (DDR) inhibitor, with an IC50 of 3.3 nM for DDR2, and shows 53% inhibition on DDR1 at 1.5 nM. |