FAAH
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB16890 | VDM 11 | 313998-81-1 | VDM 11 is a selective inhibitor of the anandamide membrane transporter (AMT) with IC50 values of 4 - 11 μM. |
| FB17732 | URB937 | 1357160-72-5 | URB937 is a FAAH inhibitor and increases anandamide levels, with an IC50 of 26.8 nM. URB937 fails to affect FAAH activity in the brain . |
| FB00790 | URB-597 | 546141-08-6 | URB-597 is fatty acid amide hydrolase (FAAH, IC50 = 4.6 nM) inhibitor without effect on other cannabinoid-related targets. |
| FB16891 | UCM 707 | 390824-20-1 | UCM 707 is an inhibitor of endocannabinoid transport and the IC50 values are 0.8 and 30 μM for the anandamide transporter and FAAH respectively. |
| FB12695 | TAK 21d | 1143578-94-2 | TAK-21d is a potent FAAH Inhibitor. |
| FB20374 | SSR 411298 | 666860-59-9 | SSR411298 is a highly selective, brain penetrant and orally-active inhibitor of FAAH with IC50 of 62.5 nM (mouse brain FAAH). |
| FB12680 | SA 47 | 792236-07-8 | SA 47 is a selective and potent inhibitor of fatty acid amide hydrolase (FAAH) and carbamate[1]. |
| FB12709 | TC-F 2 | 1304778-15-1 | Potent, reversible and selective FAAH inhibitor |
| FB12655 | SA 57 | 1346169-63-8 | Potent FAAH inhibitor |
| FB12451 | PF-750 | 959151-50-9 | PF-750 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor with IC50 of 16.2 nM. |
| FB06131 | PF-3845 | 1196109-52-0 | PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2. |
| FB01528 | PF-04457845 | 1020315-31-4 | PF-04457845 selectively inhibits FAAH with an IC50 of 7.2 nM. It has anti-inflammatory effects and is used as analgesic. |
| FB12500 | PDP-EA | 861891-72-7 | PDP-EA is an activator at FAAH. |
| FB12496 | Palmitoylisopropylamide | 189939-61-5 | Palmitoylisopropylamide is an inhibitor of fatty acid amide hydrolase (FAAH). |
| FB20323 | N-Benzyllinolenamide | 883715-18-2 | N-Benzyllinolenamide is a natural macamide isolated from Lepidium meyenii, acts as an inhibitor of fatty acid amide hydrolase (FAAH) with an IC50 of 41.8 μM. |
| FB16545 | MAFP | 188404-10-6 | MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). MAFP also binds irreversibly to CB1 receptors with IC50 of 20 nM. |
| FB05740 | LY2183240 | 874902-19-9 | LY2183240 is a highly potent blocker of anandamide uptake (IC50 = 270 pM). |
| FB02360 | JZL 195 | 1210004-12-8 | JZL195 functions as a dual inhibitor of FAAH and MAGL with IC50 of 13 nM and 19 nM respectively in brain of mouse. |
| FB02771 | JNJ-42165279 | 1346528-50-4 | JNJ-42165279 inhibits hFAAH and rFAAH with IC50 of 70 ± 8 nM and 313 ± 28 nM respectively. |
| FB01609 | JNJ-1661010 | 681136-29-8 | JNJ-1661010 is a selective inhibitor of FAAH with IC50 of 10 nM (rat) and 12 nM (human). |
| FB07828 | FAAH-IN-2 | 184475-71-6 | FAAH-IN-2 is an inhibitor of fatty acid amide hydrolase (FAAH). |
| FB08515 | FAAH Inhibitor 1 | 326866-17-5 | FAAH inhibitor 1 is a potent fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 18±8 nM. |
| FB02532 | Biochanin A | 491-80-5 | Biochanin A, a phytoestrogen from Trifolium pratense, is an inhibitor of PTK with IC50 of 91.5 μM. It also can be metabolized in vivo to genistein. |
| FB11191 | BIA 10-2474 | 1233855-46-3 | BIA10-2474 is an inhibitor of fatty acid amide hydrolase (FAAH) with IC50 of 4.9 nM. |
| FB12305 | AM 1172 | 251908-92-6 | AM 1172 is a metabolically stable anandamide uptake inhibitor (IC50 = 2.1 - 2.5 μM) and fatty acid amide hydrolase (FAAH) inhibitor (Ki = 3.18 μM). |