MAO
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB04061 | TVP1022 Mesylate | 202464-88-8 | TVP1022 mesylate is the S-isomer of rasagiline, which is an anti-Parkinson drug, appears to have the same neuroprotective activity as the R-isomer, but is 1000-fold less active as an MAO-B inhibitor. |
| FB05722 | TVP1022 | 185517-74-2 | TVP1022 is the S-isomer of rasagiline, which is an anti-Parkinson drug, appears to have the same neuroprotective activity as the R-isomer, but is 1000-fold less active as an MAO-B inhibitor. |
| FB05720 | Tranylcypromine HCl (trans) | 1986-47-6 | Tranylcypromine is a dual inhibitor of both MAO-A/B and LSD1. |
| FB08495 | Tranylcypromine Hemisulfate | 13492-01-8 | Tranylcypromine hemisulfate is an inhibitor of monoamine oxidase (MAO) and prostacyclin synthase, potently suppresses the enzymatic activity of Lysine-Specific Demethylase 1 (LSD1) (IC50 < 2 μM for BHC110/LSD1). |
| FB08809 | Tranylcypromine HCl | 4548-34-9 | Tranylcypromine HCl, is a monoamine oxidase inhibitor (MAOI) that irreversibly inhibits MAO A and MAO B with the inhibition constant Ki values of 101.9 μM and 16 μM and the half maximal inhibition concentration IC50 values of 2.3 μM and 0.95 μM respectively. |
| FB09975 | Toloxatone | 29218-27-7 | Toloxatone is an antidepressant launched in 1984 in France for the treatment of depression. |
| FB12728 | Tetrindole Mesylate | 170964-68-8 | Tetrindole was a drug candidate that functions by reversibly inhibiting monoamine oxidase A; it was first synthesized in Moscow in the early 1990s. Tetrindole is similar in its chemical structure to pirlindole (Pyrazidol), and metralindole. |
| FB10370 | TB5 | 948841-07-4 | TB5 is a potent, selective and reversible inhibitor ofhMAO-Bwith aKivalue of 0.11±0.01 μM. |
| FB11107 | Sembragiline | 676479-06-4 | Sembragiline is a selective monoamine oxidase type B inhibitor for the treatment of Alzheimer's disease. |
| FB07014 | Salsolidine | 5784-74-7 | Salsolidine is a tetrahydroisoquinoline alkaloid, acts as a stereoselective competitive MAO A inhibitor. |
| FB09367 | Safinamide Mesylate | 202825-46-5 | Safinamide mesylate is mesylate salt of safinamide, selectively and reversibly inhibits MAO-B with IC50 of 98 nM, and exhibits 5918-fold selectivity against MAO-A. |
| FB09141 | Safinamide | 133865-89-1 | Safinamide is a reversible and highly selective MAO-B inhibitor with IC50 of 98 nM. |
| FB02705 | Ro 41-1049 HCl | 127917-66-2 | Ro 41-1049 HCl is a selective, reversible, orally-active MAO-A inhibitor. |
| FB08999 | Rasagiline Mesylate | 161735-79-1 | Rasagiline Mesylate is an irreversible and selective MAO-B inhibitor used in early Parkinson's disease. |
| FB13150 | Rasagiline | 136236-51-6 | Rasagiline is an irreversible, potent and highly selective MAO-B inhibitor used to treat symptoms in early Parkinson's disease. |
| FB13150 | Rasagiline | 136236-51-6 | Rasagiline is an irreversible, potent and highly selective MAO-B inhibitor used to treat symptoms in early Parkinson's disease. |
| FB09254 | R-(-)-Deprenyl HCl | 14611-52-0 | R-(-)-Deprenyl HCl is a selective inhibitor of monoamine oxidase B (MAO-B). |
| FB08573 | Procarbazine | 671-16-9 | Procarbazine is a chemotherapy medication used for the treatment of Hodgkin's lymphoma and brain cancers. |
| FB12622 | Pirlindole Mesylate | 207572-66-5 | Pirlindole Mesylate is a highly selective reversible inhibitor of monoamine oxidase type A. |
| FB08171 | Phenelzine Sulfate | 156-51-4 | Phenelzine sulfate is a non-selective and irreversible monoamine oxidase inhibitor (MAOI), used as an antidepressant and anxiolytic. |
| FB09473 | Phenelzine | 51-71-8 | Phenelzine is a non-selective and irreversible monoamine oxidase inhibitor (MAOI), used as an antidepressant and anxiolytic. |
| FB07662 | Pargyline | 555-57-7 | Pargyline is an irreversible non-selective monoamine oxidase (MAO) inhibitor drug (IC50 for MAO-A is 11.52 nM and for MAO-B is 8.2 nM) . |
| FB08004 | Pargyline HCl | 306-07-0 | Pargyline HCl is an irreversible and selective MAO-B inhibitor with Ki values of 15 and 1.8 μM for MAO-A and MAO-B, respectively. |
| FB04234 | Paeonol | 552-41-0 | Paeonol is a naturally occuring MAO inhibitor with IC50 values of 54.6 μM and 42.5 μM for MAO-A and MAO-B, respectively. |
| FB17875 | Norharmane | 244-63-3 | Norharmane (Norharman), isolated from coffee, is a potent and selective monoamine oxidase A (MAO-A) inhibitor with a Ki of 3.34 μM. |
| FB04204 | Nialamide | 51-12-7 | Nialamide is a non-selective, irreversible monoamine oxidase inhibitor (MAOI) of the hydrazine class that was used as an antidepressant. |
| FB06313 | Mofegiline HCl | 120635-25-8 | Mofegiline HCl is a potent and selective enzyme-activated irreversible inhibitor of MAO-B and shows marked selectivity for the B form (IC50 = 680 and 3.6 nM for MAO-A and MAO-B). |
| FB08259 | Modaline Sulfate | 2856-75-9 | Modaline sulfate is a MAO inhibitor, used in the treatment of depression. |
| FB06309 | Moclobemide | 71320-77-9 | Moclobemide is a reversible MAO-A inhibitor. |
| FB04847 | Minaprine | 25905-77-5 | Minaprine is a reversible inhibitor of MAO-A, a weak inhibitor acetylcholinesterase, and an antidepressant for treatment of depression. |
| FB05944 | Minaprine 2HCl | 25953-17-7 | Minaprine 2HCl is a reversible inhibitor of MAO-A, also weakly inhibits acetylcholinesterase and is an antidepressant for treatment of depression. |
| FB04119 | Mephentermine Sulfate | 1212-72-2 | Mephentermine sulfate is a cardiac stimulant, before as a stimulant in psychiatry, has been used as a treatment for low blood pressure. |
| FB03910 | Mefexamide | 1227-61-8 | Mefexamide is a particular psychostimulant. |
| FB03344 | Lazabemide | 103878-84-8 | Lazabemide is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively). |
| FB12264 | Lazabemide HCl | 103878-83-7 | Lazabemide HCl is a selective, reversible monoamine oxidase B (MAO-B) inhibitor with IC50 of 0.03 μM. |
| FB07263 | Jatrorrhizine | 3621-38-3 | Jatrorrhizine is a protoberberine alkaloid isolated from some plant species like Enantia chlorantha. It can inhibit MAO-A and MAO-B noncompetitively with IC50 value of 4μM and 62μM, respectively. Also, it has antiinflammatory, antimicrobial and antifungal activity. |
| FB07343 | Jatrorrhizine HCl | 6681-15-8 | Jatrorrhizine HCl is a protoberberine alkaloid isolated from some plant species like Enantia chlorantha. It can inhibit MAO-A and MAO-B noncompetitively with IC50 value of 4μM and 62μM, respectively. Also, it has antiinflammatory, antimicrobial and antifungal activity. |
| FB02990 | Isatin | 91-56-5 | Isatin is an indole-derived endogenous MAO inhibitor with preferential activity against MAO-B than MAO-A. |
| FB02985 | Iproniazid Phosphate | 305-33-9 | Iproniazid Phosphate is an irreversible and non-selective MAO inhibitor. |
| FB13001 | Iproniazid | 54-92-2 | Iproniazid is an irreversible non-selective MAO inhibitor. |
| FB17851 | Hydroxyamine hydrochloride | 5470-11-1 | Hydroxyamine hydrochloride is a selective monoamine oxidase (MAO) inhibitor used for inhibiting of platelet aggregation. Hydroxyamine hydrochloride is an intermediate of organic synthesis. |
| FB10491 | Harmine | 442-51-3 | Harmine is a naturally occuring fluorescent harmala alkaloid isolated plants like Middle Eastern plant harmal which can reversibly inhibit MAOA. |
| FB09789 | Desmethoxyyangonin | 15345-89-8 | Desmethoxyyangonin is a natural kavalactones isolated and purified from the Piper methysticum (kava) plant which is an ireversible inhibitor of MAO-B. |
| FB11819 | CX157 | 205187-53-7 | CX-157 is a reversible inhibitor of monoamine oxidase-A (MAO-A) with an EC50 of 19.3 ng/mL. |
| FB07388 | Clorgiline HCl | 17780-75-5 | Clorgiline HCl is an irreversible and selective MAO-A inhibitor. |
| FB08283 | Bifemelane | 90293-01-9 | Bifemelane is a monoamine oxidase inhibitor being investigated for the treatment of depression. |
| FB12538 | Bifemelane HCl | 62232-46-6 | Bifemelane HCl is a non-selective MAO inhibitor. |
| FB07971 | Bazinaprine | 94011-82-2 | Bazinaprine is a monoamine oxidase inhibitor being investigated for the treatment of depression. |
| FB16109 | 1,4-Naphthoquinone | 130-15-4 | A choleretic. |
| FB16263 | 7-Hydroxy-3,4-dihydrocarbostyril | 22246-18-0 | 7-Hydroxy-3,4-dihydrocarbostyril is used as the materials for the organic synthesis intermediates. |