EAAT2
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB12744 | WAY 213613 | 868359-05-1 | WAY-213613 is a potent, selective GLT-1/EAAT2 (functional glutamate transporter/excitatory amino acid transporter) nonsubstrate inhibitor with IC50s of 85 nM, 5 μM and 3.8 μM for EAAT2, EAAT1 and EAAT3. WAY-213613 is a highly EAAT2-preferring transporter ligand and inhibits glutamate uptake in rat cortical synaptosomes[1][2]. |
| FB06906 | LDN-212320 | 894002-50-7 | LDN-212320 is a glutamate transporter EAAT2 activator and enhances EAAT2 levels by > 6 fold at concentrations < 5 μM after 24 h. |
| FB12731 | TFB-TBOA | 480439-73-4 | High affinity EAAT1 and EAAT2 blocker |
| FB12330 | GT 949 | 460330-27-2 | GT 949 is a potent and selective EAAT2 positive allosteric modulator with EC50 of 0.26 nM. |