SSTR
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB11231 | SSTR5 Antagonist C3p | 1628744-37-5 | SSTR5 antagonist C3p is a SSTR5 antagonist with improved PK profile and hERG inhibition activity. It can successfully exhibited a persistent glucose-lowering effect in an OGTT at a dose of 3 mg/kg. |
| FB04940 | Pasireotide L-aspartate | 396091-77-3 | Pasireotide L-aspartate is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/< 7.0/9.9 respectively). |
| FB04939 | Pasireotide | 396091-73-9 | Pasireotide is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/< 7.0/9.9 respectively). |
| FB10297 | Pasireotide Ditrifluoroacetate | 396091-75-1 | Pasireotide ditrifluoroacetate is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/< 7.0/9.9 respectively). |
| FB00207 | Octreotide | 83150-76-9 | Octreotide is an analog of somatostatin that binds to the somatostatin receptor 2/3/5. It can increase Gi activity and reduce the production of intracellular cAMP. |
| FB07825 | Octreotide Acetate | 79517-01-4 | Octreotide acetate is a long-acting octapeptide with pharmacologic actions mimicking those of the natural hormone somatostatin. |
| FB07740 | Lanreotide | 108736-35-2 | Lanreotide, a synthetic cyclic octapeptide, is the analogue of somatostatin that can inhibit somatostatin receptor 2 (SSTR-2). |
| FB09901 | Lanreotide Acetate | 127984-74-1 | Lanreotide acetate is an a synthetic cyclic octapeptide analogue of somatostatin exhibiting a high binding affinity for somatostatin receptor 2 (SSTR-2) and a lesser binding affinity for SSTR-5. |