PKA
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB04639 | Warangalone | 4449-55-2 | Warangalone is a powerful inhibitor of protein kinase A isolated and purfied from the stem bark of Erythrina addisoniae, shows marked effectiveness as an anti-inflammatory on the phospholipase A(2)-induced paw edema and on the 12-O-tetradecanoylphorbol 13-acetate-induced ear edema in mice, after systemic and local administration, respectively. |
| FB03942 | Synaptamide | 162758-94-3 | Synaptamide is a potent mediator for neurogenic differentiation of NSCs acting through PKA/CREB activation. |
| FB17715 | STAD 2 | 1542100-77-5 | STAD 2 is a PKA-tageting hydrocarbon stapled peptides. It is derived from the A Kinase Binding (AKB) domain of several AKAPs and was chemically modified to contain an all-hydrocarbon staple. Thus, it selectively binds PKA-RII and disrupt AKAP-mediated PKA signaling in cells. |
| FB12615 | PKI (5-24) | 99534-03-9 | PKI (5-24) is a high affinity PKA inhibitor with Ki of 2.3 nM. |
| FB02206 | H 89 | 127243-85-0 | H 89 is a potent and selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A) with IC50 of 48 nM showing weak inhibition on PKG, PKC, CK1, CK2 and others kinases. |
| FB10148 | H 89 2HCl | 130964-39-5 | H 89 2HCl is a potent and selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A) with IC50 of 48 nM. It also shows weak inhibition on PKG, PKC, CK1, CK2 and others kinases. |
| FB12122 | GSK180736A | 817194-38-0 | GSK180736A is an inhibitor of G protein-coupled receptor kinase 2 (GRK2) with IC50 of 0.77 μM. |
| FB08847 | Dibutyryl-cAMP | 16980-89-5 | Dibutyryl-cAMP inhibits neuronal glucose uptake via PKA activation. |
| FB12207 | CW 008 | 1134613-19-6 | CW 008 is a PKA signaling activator. |
| FB06976 | Bucladesine Calcium | 938448-87-4 | Bucladesine Calcium is a cell-permeable PKA activator that functions by preferentially activating endogenous cAMP. |
| FB07106 | 8-Bromo-cAMP | 76939-46-3 | 8-Bromo-cAMP is a cell permeable analog of cAMP that activates cyclic-AMP-dependent protein kinase with a Ka value of 0.05 μM and a PKA activator. |