CAS:204067-01-6PD176252

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PD176252 PD176252 Cat No. FB11749Cas No. 204067-01-6

PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells.

规格	价格	促销价格	库存

18817579266

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18817579266

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实验数据

储存液制备
- 1 mg
- 5 mg
- 10 mg
- 1 mM
- 1.7104 mL
- 8.5519 mL
- 17.1038 mL
- 5 mM
- 0.3421 mL
- 1.7104 mL
- 3.4208 mL
- 10 mM
- 0.1710 mL
- 0.8552 mL
- 1.7104 mL
计算器摩尔计算器总药量计算器工作液计算器

技术信息

CAS号	204067-01-6	储存条件	粉末 -20°C 3 年液体 -80°C 12 月
分子式	C32H36N6O5	运输	蓝冰
分子量	584.67	别名

靶点数据

生物活性

描述PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells.