EZH2 (stapled peptide) refers the stapled peptide target EZH2.
货号 | 产品名 | CAS号 | 信息 |
---|---|---|---|
FB17710 | SAH-EZH2 | 1453222-26-8 | SAH-EZH2 is a EZH2-targeting stapled peptide that selectively inhibits H3 Lys27 trimethylation by dose-responsively disrupting the EZH2/EED complex and reducing EZH2 protein levels, a mechanism distinct from that reported for small molecule EZH2 inhibitors targeting the enzyme catalytic domain. |