Adenosine Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| FB01167 | ZM241385 | 139180-30-6 | ZM241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor. |
| FB05312 | Tubotaiwine | 6711-69-9 | Tubotaiwine, a natural product isolated and purified from the herbs of Ervatamia divaricata, shows selective activity against L. infantum., and has affinity for adenosine receptors in the micromolar range and also have in-vivo analgesic activity in mice. |
| FB03058 | Tozadenant | 870070-55-6 | Tozadenant is a selective adenosine A2A receptor antagonist with Ki values of 11.5 nM on human A2A and 6 nM on rhesus A2A, which can improve motor function in animal models of Parkinson's disease. |
| FB09209 | SCH-58261 | 160098-96-4 | SCH 58261 is a potent and selective A2a adenosine receptor antagonist with Ki of 2.3 nM and 2 nM for rat A2a and bovine A2a, respectively. |
| FB08790 | Regadenoson | 313348-27-5 | Regadenoson is a selective adenosine A2A receptor agonist with Ki value of 1.1nM for pig striatum A2A receptor, used as a novel pharmacologic stress agent under clinical development for myocardial perfusion imaging. |
| FB08645 | Propentofylline | 55242-55-2 | Propentofylline, a xanthine derivative with purported neuroprotective effects, acts as a c-AMP phosphodiesterase inhibitor, a nerve growth factor stimulator, an adenosine transport inhibitor and a non-selective adenosine receptor antagonist. |
| FB02861 | Preladenant | 377727-87-2 | Preladenant is a highly selective and competitive A2A receptor antagonist with Ki value of 1.1nM, used in trials studying the treatment of brain diseases, such as parkinson disease, movement disorders, antipsychotic agents and parkinsonian disorders. |
| FB03469 | PD117519 | 96392-15-3 | PD117519 is an adenosine agonist. |
| FB07121 | N6-Cyclohexyladenosine | 36396-99-3 | N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). |
| FB02656 | Istradefylline | 155270-99-8 | Istradefylline is a very potent, selective and orally active adenosine A2A receptor antagonist (Ki=2.2 nM) in experimental models of Parkinson's disease. |
| FB01306 | Enprofylline | 41078-02-8 | Enprofylline is a xanthine derivative used in the treatment of asthma, which acts as a bronchodilator. |
| FB09397 | CGS 21680 | 120225-54-9 | CGS 21680 is an adenosine A2 receptor agonist with IC50 of 22 nM, exhibits 140-fold over A1 receptor. |
| FB09168 | Capadenoson | 544417-40-5 | Capadenoson is an oral active, potent and selective adenosine A1 receptor agonist. |
| FB07823 | Acefylline | 652-37-9 | Acefylline is an adenosine receptor antagonist, a stimulant drug of the xanthine chemical class. |
| FB12565 | 1,3-Dipropyl-8-phenylxanthine | 85872-53-3 | |
| FB12782 | PSB 1115 | 152529-79-8 |