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Synonyms: LS190926
XE991 is a potent and selective blocker of KV7 (KCNQ) voltage-gated potassium channels which blocks KV7.2+7.3 (KCNQ2+3) / M-currents (IC50 = 0.6 - 0.98 μM) and KV7.1 (KCNQ1) homomeric channels (IC50 = 0.75 μM) but is less potent against KV7.1/minK channels (IC50 = 11.1 μM).
规格 | 价格 | 促销价格 | 库存 |
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18817579266
实验数据
技术信息
CAS号 | 122955-42-4 | 储存条件 |
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分子式 | C26H20N2O | 运输 | 蓝冰 | |
分子量 | 376.45 | 别名 | LS190926 |
生物活性