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UK-78282 is a blocker of the KV1.3 and KV1.4 voltage-gated potassium channels in T lymphocytes (IC50 values are 0.28 and 0.17 μM respectively) which suppresses T lymphocyte mitogenesis and leads to membrane depolarization and also blocks KV1.4 expressed in heart and brain.
规格 | 价格 | 促销价格 | 库存 |
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18817579266
实验数据
技术信息
CAS号 | 136647-02-4 | 储存条件 |
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分子式 | C29H36ClNO2 | 运输 | 蓝冰 | |
分子量 | 466.06 | 别名 |
生物活性