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UB-165 is a potent nAChR ligand, which displays functional selectivity between nAChR subtypes. It is a full agonist at α3β2- and very weak partial agonist at α4β2- containing nAChRs with Ki values of 0.27, 20 (IC50), 2790 and 990 nM for α4β2, α3, α7 and α1β1δε respectively.
规格 | 价格 | 促销价格 | 库存 |
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18817579266
实验数据
技术信息
CAS号 | 2454492-43-2 | 储存条件 |
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分子式 | C17H19ClN2O4 | 运输 | 蓝冰 | |
分子量 | 350.80 | 别名 |
生物活性