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PI-103 is a potent inhibitor with low IC50 values against recombinant PI3K isoforms p110alpha (IC50= 2 nM), p110beta (IC50= 3 nM), p110delta (IC50= 3 nM), and p110gamma (IC50= 15 nM), less potent to mTOR/DNA-PK with IC50 of 30 nM/23 nM.
规格 | 价格 | 促销价格 | 库存 |
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18817579266
实验数据
技术信息
CAS号 | 371935-74-9 | 储存条件 |
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分子式 | C19H16N4O3 | 运输 | 蓝冰 | |||||||||||||
分子量 | 348.36 | 别名 | ||||||||||||||
溶解度 |
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动物实验配方 |
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靶点 | Description | IC50 |
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DNA-PK | IC50:23nM | |
mTOR | IC50:30nM | |
p110α | IC50:2nM | |
p110β | IC50:3nM | |
p110γ | IC50:15nM | |
p110δ | IC50:3nM |