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Synonyms: 9-Bromopaullone;NSC-664704
Kenpaullone is an ATP-competitive inhibitor of CDK1/cyclin B (IC50 = 0.4 µM), CDK2/cyclin A (IC50 = 0.68 µM), CDK5/p25 (IC50 = 0.85 µM), lymphocyte kinase (IC50 = 0.47 µM) , and GSK-3β (C50 = 0.23 μM).
规格 | 价格 | 促销价格 | 库存 |
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18817579266
实验数据
技术信息
CAS号 | 142273-20-9 | 储存条件 |
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分子式 | C16H11BrN2O | 运输 | 蓝冰 | |||||||||||
分子量 | 327.18 | 别名 | 9-Bromopaullone;NSC-664704 | |||||||||||
溶解度 |
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动物实验配方 |
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生物活性
靶点 | GSK-3β IC50:0.23μM | Lck IC50:0.47μM | CDK2/cyclin A IC50:0.68μM | CDK5/p25 IC50:0.85μM |
靶点 | Description | IC50 |
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GSK-3β | IC50:0.23μM | |
Lck | IC50:0.47μM | |
CDK2/cyclin A | IC50:0.68μM | |
CDK5/p25 | IC50:0.85μM |