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Synonyms: CHIR-99021 HCl
CHIR-99021 HCl is HCl of CHIR-99021, which is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM and shows greater than 500-fold selectivity for GSK-3 versus its closest homologs Cdc2 and ERK2.
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18817579266
实验数据
技术信息
CAS号 | 1797989-42-4 | 储存条件 |
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分子式 | C22H19Cl3N8 | 运输 | 蓝冰 | |||||||||
分子量 | 501.80 | 别名 | CHIR-99021 HCl | |||||||||
溶解度 |
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动物实验配方 |
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生物活性