产品
编 号:F146987
分子式:C22H30N4O4S
分子量:446.56
产品类型
结构图
CAS No: 1388896-07-8
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生物活性:
ND-2158 is a competitive IRAK4 inhibitor, with the Ki of 1.3 nM. ND-2158 suppresses LPS-induced TNF production in human white blood cells, alleviated collagen-induced arthritis, and blocked gout formation in mouse models. ND-2158 has antitumor activity in vivo.