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编 号:F124654
分子式:C17H19FN2O2
分子量:302.34
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10mM*1mL in DMSO
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5mg
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10mg
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50mg
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生物活性:
Ralfinamide (FCE-26742A) is an orally available Na+ blocker derived from α-aminoamide, with function of suppressing pain.

体内研究:
Ralfinamide (30 mg/kg, 60 mg/kg; p.o.; twice daily; 42 days) treated with Ralfinamide (80 mg/kg; p.o.; twice daily; 7 days) preoperatively suppresses neuropathic pain.Animal Model:81 adult male Sprague–Dawley male rats (260–460 g)
Dosage:80 mg/kg (7 days preoperatively), 30 mg/kg, 60 mg/kg (postoperative)
Administration:Oral gavage; twice daily; until postoperative day 42
Result:Suppressed neuropathic pain.
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