产品
编 号:F763010
分子式:C49H53ClFN5O5
分子量:846.43
产品类型
结构图
CAS No: 3031307-73-7
联系客服
产品详情
生物活性:
EGFR-IN-42 (Compound 17b) is a potent inhibitor of EGFR with single-digit nanomolar activity. EGFR-IN-42 connects tamoxifen or endoxifen with the EGFR-inhibitor gefitinib via a covalent linkage. EGFR-IN-42 retains both ER antagonist activity and EGFR inhibition. EGFR-IN-42 has superior anti-cancer activity.