产品
编 号:F762376
分子式:C22H28N6O4
分子量:440.5
产品类型
结构图
CAS No: 1809163-24-3
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产品详情
生物活性:
HDAC-IN-43 is a potent HDAC 1/3/6 inhibitor with IC50 values of 82, 45, and 24 nM, respectively. HDAC-IN-43 is a weak PI3K/mTOR inhibitors with IC50 values of 3.6 and 3.7 μM, respectively. HDAC-IN-43 shows broad anti-proliferative activity .
体外研究:
HDAC-IN-43 demonstrats broad anti-cancer activities against 38 cancer cell lines at 72 hours .