产品
编 号：F083986
分子式：C17H21Cl2N3O3
分子量：386.27
分子式：C17H21Cl2N3O3
分子量：386.27
产品类型
规格
价格
是否有货
5mg
300
In-stock
10mg
480
In-stock
50mg
1680
In-stock
100mg
2880
In-stock
结构图
CAS No: 123040-16-4
产品详情
生物活性：
Azasetron (Y-25130) hydrochloride, a benzamide derivative, is a potent and selective 5-HT3 receptor antagonist. Azasetron is used in the study for Chemotherapy-induced nausea and vomiting (CINV).
体内研究：
Azasetron could effectively penetrate through the skin and pass into the systemic circulation.Animal Model:Four male Bama miniature pigs weighing 9-11 kg (15-16 weeks old).
Dosage:0.5 mg/kg.
Administration:I.V. administration via the abdominal vein.
Result:The mean plasma concentration dropped to minimum at 36 h. Cmax = 44.88 ± 7.16 ng/mL) was achieved at the time point of 66.00 ± 22.98 h (Tmax).
Azasetron (Y-25130) hydrochloride, a benzamide derivative, is a potent and selective 5-HT3 receptor antagonist. Azasetron is used in the study for Chemotherapy-induced nausea and vomiting (CINV).
体内研究：
Azasetron could effectively penetrate through the skin and pass into the systemic circulation.Animal Model:Four male Bama miniature pigs weighing 9-11 kg (15-16 weeks old).
Dosage:0.5 mg/kg.
Administration:I.V. administration via the abdominal vein.
Result:The mean plasma concentration dropped to minimum at 36 h. Cmax = 44.88 ± 7.16 ng/mL) was achieved at the time point of 66.00 ± 22.98 h (Tmax).
产品资料
Copyright©2015-2024 沪ICP备2022026524号-1
沪公网安备