产品
编 号:F083130
分子式:C22H24ClN5O
分子量:409.91
产品类型
结构图
CAS No: 1228088-30-9
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产品详情
生物活性:
Balovaptan (RG7314) is an orally available, selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors, and is used for the research of autism.
体外研究:
Balovaptan (RG7314) shows >30000-fold selectivity for hV1a over hV2 receptors, 9891-fold selectivity over hOTR (human oxytocin receptor).