产品
编 号:F759335
分子式:C30H40N6O6S
分子量:612.74
产品类型
结构图
CAS No: 63307-63-1
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产品详情
生物活性:
(D-Met2,Pro5)-Enkephalinamide is a highly potent opiate agonist, and shows antinociceptive activity.
体内研究:
(D-Met2,Pro5)-Enkephalinamide (intravenous injection; 0.25 and 0.5 mg/kg; once) leads to the decreasement of prolactin (PRL) secretion in lactating rats.Animal Model:Wistar lactating rats
Dosage:0.25 and 0.5 mg/kg
Administration:Intravenous injection; 0.25 and 0.5 mg/kg; once
Result:Decreased plasma PRL levels 15 min after the administration in continuously lactating rats.Produced a marked depression in plasma PRL concentration in non-deprived lactating mothers.