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编 号:F758924
分子式:C21H26BrNO3
分子量:420.34
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生物活性:
Parapenzolate bromide, an antispasmodic, is an orally active mAChR antagonist. Parapenzolate bromide is an anticholinergic agent.

体内研究:
Parapenzolate bromide (10 mg/kg, p.o. or i.v.) shows a significant analgesic effect in mice.Parapenzolate bromide (0.5 mg/kg, i.v.) exhibits a spasmolytic activity in isolated gall bladder from guinea pigs.Animal Model:Mice
Dosage:10 mg/kg
Administration:Oral administration (p.o.) or intravenous injection (i.v.)
Result:Prolonged the time until death in convulsive mice.
Animal Model:Guinea pigs
Dosage:0.5 mg/kg
Administration:Intravenous injection (i.v.)
Result:Antagonized contractions induced by acetylcholine (100 μg/kg, i.v.)
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