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编 号:F756932
分子式:C24H23N7O2
分子量:441.49
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结构图
CAS No: 2924182-31-8
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生物活性:
PHD-IN-1 (compound 80) is a potent inhibitor of PHD2,with an IC50 value of ≤5 nM. PHD-IN-1 shows EC50s of 2.5 μM in EPO Elisa assay both in Caco2-HIFla-HiBiT-clone-1 cells and Hep3B cells,respectively.