产品
编 号:F756651
分子式:C49H73N13O11
分子量:1020.18
产品类型
结构图
CAS No: 2891469-81-9
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产品详情
生物活性:
NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal) (compound 40), a macrocyclic analogue of Ape13, is a potent APJ agonist (Ki=5.7 nM). NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal) exhibits a favorable Gα12-biased signaling and an increased in vivo half-life.