产品
编 号:F756550
分子式:C26H23F3N6
分子量:476.5
产品类型
结构图
CAS No: 2878441-72-4
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产品详情
生物活性:
USP1-IN-4 (compound 10) is an effective USP1 inhibitor with an IC50 value of 2.44 nM. USP1-IN-4 has anticancer activity and synergistic activity with various anticancer drugs.
体外研究:
USP1-IN-4 (0.0005-10 μM, 15 分钟) 显著抑制USP1/UAF1,IC50 为 2.44 nM。USP1-IN-4 (0.0005-10 μM, 7 天) 显著抑制MDA-MB-436生长,IC50 为 103.75 nM。