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编 号:F755190
分子式:C29H38IN5
分子量:583.55
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结构图
CAS No: 2743448-32-8
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Dim16 is a dual PCSK9/HMG-CoAR inhibitor, with an IC50 value of 19 nM for PCSK9. Dim16 inhibits PCSK9-LDLR binding with an IC50 value of 0.8 nM. Dim16 increases LDL uptake in HepG2 cells.