产品
编 号:F754724
分子式:C27H31NO3
分子量:417.54
产品类型
结构图
CAS No: 2699724-40-6
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生物活性:
(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma.