产品
编 号:F754601
分子式:C49H59ClN8O8S2
分子量:987.62
产品类型
规格
价格
是否有货
10mM*1mL in DMSO
询价
询价
1mg
询价
询价
5mg
询价
询价
结构图
联系客服
产品详情
生物活性:
OARV-771 is a VHL-based BET degrader (PROTAC) with improved cell permeability. OARV-771 shows DC50s of 6, 1, and 4 nM for Brd4, Brd2 and Brd3, respectively.

体外研究:
OARV-771 shows antiproliferative effect with an EC50 value of 4 nM in MV4;11.
产品资料