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编 号:F753131
分子式:C13H7Cl2NO3S
分子量:328.17
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生物活性:
CAXII-IN-1 (Compound 17) is a selective CA XII inhibitor with Ki values of 3.8 nM and 56.0 nM against hCA XII and hCA IX, respectively. CAXII-IN-1 shows antitumor activity.

体外研究:
CAXII-IN-1 (Compound 17) shows cytotoxicity with IC50 values of 20±1, 4.8±0.03 and 14±2 μM against MCF-7, HeLa and A549 cells, respectively.
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