产品
编 号:F751613
分子式:C57H68FN11O8S
分子量:1086.28
产品类型
结构图
CAS No: 2374122-43-5
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产品详情
生物活性:
PROTAC IRAK4 degrader-3 is a PROTAC-induced IRAK4 degrader based on von Hippel-Lindau.
体外研究:
PROTAC IRAK4 degrader-3 (0.01~10 μM; 2 hours; PBMCs) mediated degradation is occurring in a proteasome dependent manner.PROTAC IRAK4 degrader-3 (0.01~100 μM; 18 hours; PBMCs) is capable of completely blocking IL-6 secretion.