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编 号:F751320
分子式:C52H66N2O20P2
分子量:1101.03
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生物活性:
Pomstafib-2 is a potent and selective STAT5b inhibitor. Pomstafib-2 decreases the expression of pSTAT5b and induces Apoptosis.

体外研究:
Pomstafib-2 (compound 8) (0-10 μM; 4 h) decreases the expression of pSTAT5b in a dose-dependent manner in STAT5b-GFP-transfected K562 cells.Pomstafib-2 (0, 10, 20, 40, 60, 80 μM; 48 h) induces apoptosis in a dose-dependent manner in STAT5-dependent K562 cells.
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