产品
编 号:F751081
分子式:C12H13ClF3N
分子量:263.69
产品类型
结构图
CAS No: 230615-01-7
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产品详情
生物活性:
(Rac)-CP-601927 hydrochloride is the racemate of CP-601927. CP-601927 is a nAChR agonist with Ki values 1.2 nM and 102 nM for α4β2 and α3β4 nAChR, respectively.
体外研究:
CP-601927 induces significant antidepressant-like effects in mice. CP-601927 could decrease cholinergic signaling as a result of its reduced efficacy or via desensitization of α4β2* nAChRs.