产品
编 号:F749984
分子式:C19H20FNO4S
分子量:377.43
产品类型
结构图
CAS No: 2226732-62-1
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产品详情
生物活性:
CVN636 is a potent, orally active and selective mGluR7 allosteric agonist with an EC50 value of 7 nM for hu mGluR7. CVN636 has central nervous system (CNS) permeability.
体内研究:
CVN636 (0.3-3 mg/kg; p.o.) 减少 msP 大鼠的乙醇自我给药。Animal Model:msP rat
Dosage:0.3, 1, and 3 mg/kg
Administration:oral administration
Result:Reduced alcohol self-administration in a dose-dependent.