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编 号:F749571
分子式:C25H24F4N2O2
分子量:460.46
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结构图
CAS No: 2170766-56-8
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生物活性:
Estrogen receptor modulator 8 (compound 4) is an orally active inhibitor of Estrogen Receptor/ERR α (IC50=0.437 nM, MCF-7 cells). Estrogen receptor modulator 8 inhibits MCF-7 cells proliferation with an IC50 value of 0.1 nM.