产品
编 号:F749169
分子式:C20H18FNO3
分子量:339.36
产品类型
结构图
CAS No: 2126784-39-0
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产品详情
生物活性:
VU6010572 is a potent and selective mGlu3 negative allosteric modulator with IC50 of 245 nM. VU6010572 is highly CNS penetrant.
体内研究:
VU6010572 (3 mg/kg; i.p.) shows robust efficacy.VU6010572 (3 mg/kg; i.p.; 45 minutes) produces lasting anxiolytic-like behavioral effects.Animal Model:CD-1 mice
Dosage:3 mg/kg
Administration:I.p.
Result:Showed robust efficacy.
Animal Model:Rats
Dosage:3 mg/kg
Administration:I.p.; 45 minutes
Result:Produced lasting anxiolytic-like behavioral effects.