产品
编 号:F749094
分子式:C21H32N2O5S
分子量:424.55
产品类型
结构图
CAS No: 2114324-48-8
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生物活性:
Danavorexton (TAK-925) is an orexin receptor agonist with brain permeability. Danavorexton induces a physiological pattern of OX2R activation in vitro to wake up sleepy mice and improve sleepiness symptoms.
体内研究:
Danavorexton (1, 10 mg/kg 或1, 3 mg/kg, 皮下注射) 剂量依赖性增强了普通狨猴和食蟹猴的觉醒。Animal Model:Common marmosets and cynomolgus monkeys models
Dosage:1, 10 mg/kg (1, 3 mg/kg)
Administration: s.c.
Result:Decreased SWS I (Sleeping With Sirens I), SWS II (Sleeping With Sirens II) and REM (Rapid Eye Movement) sleep time.