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编 号:F748912
分子式:C23H22N4O3
分子量:402.45
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生物活性:
TP-030-1 is an inhibitor of RIPK1. TP-030-1 inhibits hRIPK1 with a Ki value of 3.9 nM and inhibits mRIPK1 with an IC50 value of 4.2 μM. TP-030-1 can be used for the research of inflammatory diseases and neurodegenerative diseases.

体外研究:
TP-030-1 inhibits HT29 necroptosis with an IC50 value of 18 nM.TP-030-1 inhibits hRIPK1 with a Ki value of 3.9 nM.TP-030-1 inhibits mRIPK1 with an IC50 value of 4.2 μM.
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