产品
编 号:F747812
分子式:C19H15Cl2NO3
分子量:376.23
产品类型
结构图
CAS No: 1903783-77-6
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产品详情
生物活性:
(+)-TK216 is an enantiomer of TK216 (HY-122903). TK216 is an orally active and potent E26 transformation specific (ETS) inhibitor.
体外研究:
(+)-TK216 (compound 13; for 3 days) has an IC50>5 μM in SKES cells (Ewing Sarcoma cell line). (+)-TK216 has T1/2s of 103.4 mins, 3.6 mins, 26.6 mins and 8.4 mins for human, rat, mouse, dog liver microsomes.