产品
编 号：F747245
分子式：C18H25N3O2
分子量：315.41
分子式：C18H25N3O2
分子量：315.41
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规格
价格
是否有货
结构图
CAS No: 1808463-81-1
产品详情
生物活性：
GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with an Ki of 0.56 μM. GABAA receptor agent 6 shows γ-GABAAR antagonist activity with low cellular membrane permeability.
体外研究：
GABAA receptor agent 6 (compound 2027) shows antagonist activity with IC50s of 6.68, 1.03, 0.36, 4.13, 4.96, 2.96, 0.29, 0.59 μM for α1β2δ, α4β1δ, α4β2δ, α6β2δ, α1β2γ2, α2β2γ2, α3β2γ2, α5β2γ2 subtypes, respectively.
GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with an Ki of 0.56 μM. GABAA receptor agent 6 shows γ-GABAAR antagonist activity with low cellular membrane permeability.
体外研究：
GABAA receptor agent 6 (compound 2027) shows antagonist activity with IC50s of 6.68, 1.03, 0.36, 4.13, 4.96, 2.96, 0.29, 0.59 μM for α1β2δ, α4β1δ, α4β2δ, α6β2δ, α1β2γ2, α2β2γ2, α3β2γ2, α5β2γ2 subtypes, respectively.
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