产品
编 号:F747184
分子式:C34H43N3O8
分子量:621.72
产品类型
结构图
CAS No: 1803040-07-4
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产品详情
生物活性:
20S Proteasome-IN-3 is a 20S proteasome β5 subunit inhibitor (IC50=1.64 μM). 20S Proteasome-IN-3 shows anti-tumor proliferation activity.
体外研究:
20S Proteasome-IN-3 (Compound 10b) (5.34-9.69 μM, 18-24 h) exhibits significant inhibition against A375, SW480, DU145, and HeLa cells.