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编 号:F746340
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CAS No: 1629605-31-7
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生物活性:
Domagrozumab is an anti-myostatin humanized monoclonal antibody with a KD value of 2.6 pM for human myostatin. Domagrozumab induces muscle anabolic activity. Domagrozumab can be used in research of duchenne muscular dystrophy (DMD).
体内研究:
Domagrozumab (PF-06252616; 10 and 30 mg/kg; i.v.) 以剂量依赖性方式增加肌肉生长抑制素水平并诱导食蟹猴骨骼肌肥大。
体外研究:
Domagrozumab (PF-06252616) 抑制人肌肉生长抑制素信号传导活性,IC50 值 为 Domagrozumab 相关抗体: